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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T5449 | Bamaquimast | L 0042,F 10126 | Proton pump |
Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system disorders and respiratory diseases. | |||
T10152 | 4-Methylamino antipyrine | COX , Drug Metabolite | |
4-Methylamino antipyrine is an active metabolite of Metamizole. Metamizole is a pyrazolone non-steroidal anti-inflammatory drug (NSAID) and inhibits COX. 4-Methylamino antipyrine has analgesic, antipyretic, and relativel... | |||
T4561 | Tiaprofenic acid | Tiaprofensaeure,Acido tiaprofenico,Surgam | Others , COX |
Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain. | |||
T36683 | Vedaprofen | Quadrisol,PM 150,CERM 10202 | COX , Antibacterial , Prostaglandin Receptor |
Vedaprofen (PM 150) inhibits COX-1 and reduces prostaglandin H2 synthesis with anti-inflammatory activities. Vedaprofen is an inhibitor of Escherichia coli sliding clamp with the IC50 of 222 μM and Ki of 131 μM. | |||
T50025 | Lonazolac | PPAR | |
Lonazolac is a nonsteroidal anti-inflammatory drug[1]. | |||
T6540 | Ibuprofen Lysine | Neoprofen | COX |
Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug. | |||
T0258 | Carsalam | Carsalame,Carbonylsalicylamide,2H-1,3-Benzoxazine-2,4(3H)-dione | Antibiotic |
Carsalam (2H-1,3-Benzoxazine-2,4(3H)-dione) is a nonsteroidal anti-inflammatory drug. | |||
T0321 | Indoprofen | (±)-Indoprofe | COX |
Indoprofen ((±)-Indoprofe) is a non-steroidal anti-inflammatory drug. | |||
T19679 | Benoxaprofen | NSC 299582,LY-90459,Benoxaphen. Compound 90459 | COX |
Benoxaprofen (NSC-299582) is a non-steroidal anti-inflammatory drug. | |||
T1421 | Aceclofenac | Preservex,Airtal | COX |
Aceclofenac (Preservex) is a non-steroidal anti-inflammatory drug (NSAID) with marked anti-inflammatory and analgesic properties. | |||
T1280 | Nepafenac | AL 6515,AHR 9434 | COX |
Nepafenac (AHR 9434) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of nepafenac is as a Cyclooxygenase Inhibitor. The chemical classification of nepafenac is Nonsteroidal Anti-inflammatory Compounds. | |||
T6498 | Fenoprofen calcium hydrate | Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate | Apoptosis , Others , COX |
Fenoprofen calcium hydrate (Progesic dihydrate) is a non-steroidal anti-inflammatory drug (NSAID). | |||
T19636 | Morniflumate | Niflam,UP 164,UP-164,Morniflu,UP164 | Others |
Morniflumate (Niflam) is a nonsteroidal anti-inflammatory drug. It is used to treat inflammation. | |||
T11340 | Furprofen | Prostaglandin Receptor | |
Furprofen, a non-steroidal anti-inflammatory drug (NSAID), exerts its effects by inhibiting the synthesis of prostaglandin (PGE). This compound demonstrates analgesic properties and can be conveniently administered orall... | |||
T6387 | Ampiroxicam | CP 65703,Flucam | COX |
Ampiroxicam (Flucam) is a nonselective cyclooxygenase inhibitor uesd as anti-inflammatory drug. | |||
T20615 | Olsalazine | Dipentium,Salicylic acid | Others |
Olsalazine (Dipentium), an anti-inflammatory drug, is used in the treatment of inflammatory bowel disease. It is also a novel DNA hypomethylating agent. | |||
T0310 | Actarit | 4-acetylaminophenylacetic acid | Others |
Actarit (4-acetylaminophenylacetic acid) is an anti-inflammatory drug. | |||
T0826 | Meloxicam | Movalis,Mobic,Metacam | Apoptosis , COX , Autophagy |
Meloxicam (Metacam) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of meloxicam is as a Cyclooxygenase Inhibitor. The chemical classification of meloxicam is Nonsteroidal Anti-inflammatory Compounds. | |||
T2550 | Tolmetin | Tolectin | COX |
Tolmetin (Tolectin) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of tolmetin is as a Cyclooxygenase Inhibitor. The chemical classification of tolmetin is Nonsteroidal Anti-inflammatory Compounds. | |||
T1582 | Naproxen | (S)-Naproxen | COX , Autophagy |
Naproxen ((S)-Naproxen) is a propionic acid derivative and a non-steroidal anti-inflammatory drug (NSAID) with anti-inflammatory, antipyretic and analgesic activities. | |||
T1720 | Amfenac Sodium Hydrate | Amfenac Sodium Monohydrate | COX |
Amfenac Sodium Hydrate is a non-steroidal analgesic anti-inflammatory drug with acetic acid moiety. | |||
T3608 | Carbasalate calcium | Rheomin,Omegin,Alcacyl,Iromin,Solupsan,Carbasalate Calcium | Platelet aggregation |
Carbasalate calcium (Rheomin) is an analgesic, antipyretic, and anti-inflammatory drug, as well as a platelet aggregation inhibitor. | |||
T1325 | Carprofen | Ridamyl,Imadyl,Rimadyl | FAAH , COX , Autophagy |
Carprofen (Ridamyl) is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic activities. | |||
T0319 | Suxibuzone | Calibene,Suxibuzonum,Suxibuzona | COX |
Suxibuzone (Suxibuzona) is a drug used for joint and muscular pain. It is a prodrug of the non steroidal anti inflammatory drug phenylbutazone, and is commonly used in horses. | |||
T0708 | Oxaprozin | Oxaprozinum,Wy21743 | NF-κB , COX |
Oxaprozin (Oxaprozinum) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of oxaprozin is as a Cyclooxygenase Inhibitor. The chemical classification of oxaprozin is Nonsteroidal Anti-inflammatory Compound... | |||
T0466 | Celecoxib | SC 58635 | COX |
Celecoxib (SC 58635) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of celecoxib is as a Cyclooxygenase Inhibitor. | |||
T4966 | Ufenamate | Flufenamic acid butyl ester,Butyl flufenamate | Others |
Ufenamate (Flufenamic acid butyl ester) is an anthranilic acid-based anti-inflammatory drug developed for skin diseases | |||
T0498 | Salsalate | Disalicylic acid,Salicylsalicylic acid,Sasapyrine,NSC-49171 | Reactive Oxygen Species , COX |
Salsalate (Sasapyrine) is an orally available salicylate and non-steroidal anti-inflammatory drug (NSAID), with anti-inflammatory, analgesic and antipyretic activities. | |||
T23403 | Sulindac sulfone | Reductase , COX | |
Sulindac sulfone is a metabolite of the nonsteroidal anti-inflammatory drug sulindac. | |||
T7882 | Indomethacin farnesil | Infree | Others , COX , Autophagy |
Indomethacin farnesil (Infree) is a prodrug of indomethacin. It acts as a nonsteroidal anti-inflammatory drug (NSAID) and disease-modifying anti-rheumatic drug (DMARD). | |||
T1258 | Nabumetone | BRL14777 | COX , Glutathione Peroxidase |
Nabumetone (BRL14777)(BRL14777) is a non-steroidal anti-inflammatory drug and its active metabolite 6MNA inhibits the enzymes cyclo-oxygenase I and II. | |||
T4542 | Clonixin | Clonixic acid | Others |
Clonixin (Clonixic acid) is a non-steroidal anti-inflammatory drug (NSAID) with analgesic properties. This compound has been reported to block prostaglandin synthesis, and to block inward calcium currents. | |||
T0448 | (S)-(+)-Ibuprofen | Dexibuprofen,(S)-Ibuprofen | BCL , Thrombin , Cysteine Protease , COX , PPAR |
(S)-(+)-Ibuprofen (Dexibuprofen) , is a non-steroidal anti-inflammatory drug (NSAID), inhibiting cyclooxygenase (COX). | |||
T6424 | Bromfenac Sodium | AHR 10282B,Bronuck,AHR 10282R | COX |
Bromfenac Sodium (AHR 10282R) is a nonsteroidal anti-inflammatory drug (NSAID), which has anti-inflammatory activity and may block prostaglandin synthesis by inhibiting cyclooxygenase 1 and 2. | |||
T0159 | Pranoprofen | Pyranoprofen | Apoptosis , COX , PGE Synthase , Prostaglandin Receptor |
Pranoprofen (Pyranoprofen) (INN) is a non-steroidal anti-inflammatory drug used in ophthalmology. | |||
T0055 | Glafenine | Glafenin | COX |
Glafenine (Glafenin), a non-narcotic analgesic agent, is a non-steroidal anti-inflammatory drug (NSAID), and widely used for the therapy of pains of various origins. | |||
T1394 | Ibuprofen | Brufen,(±)-Ibuprofe,Motrin,Advil | COX |
Ibuprofen (Advil) is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic effects. Ibuprofen inhibits the activity of cyclo-oxygenase I and II, resu... | |||
T0285 | Isoxicam | Isoxicamum,Isoxicamo,Maxicam | COX |
Isoxicam (Isoxicamum) is a non-steroidal anti-inflammatory drug that is not marketed in the United States. | |||
T1191L | Metamizole sodium | Analgin,Dipyron | COX |
Metamizole sodium (Analgin) is a drug that has analgesic, anti-inflammatory, and antipyretic properties. It is the sodium sulfonate of AMINOPYRINE. | |||
T0726 | Benzydamine hydrochloride | Benzydamine HCl,AF864 | COX , PGE Synthase , Antibacterial |
Benzydamine hydrochloride (AF864), a locally-acting nonsteroidal anti-inflammatory drug, has local anaesthetic and analgesic properties. | |||
T0767 | Sulfapyridine | Sulfidine,Sulfidin,2-Sulfapyridine | Antibacterial , Antibiotic , Autophagy |
Sulfapyridine (2-Sulfapyridine) is a short-acting sulfonamide antibiotic and by-product of the non-steroidal anti-inflammatory drug sulfasalazine. | |||
T21412 | Ketorolac | Toradol,Sprix,Acuvail,Macril,Acular | COX |
Ketorolac (Acuvail) is a non-steroidal anti-inflammatory drug (NSAID) in the family of heterocyclic acetic acid derivatives. It acts by inhibiting the bodily synthesis of prostaglandins. | |||
T28972 | Tiaramide hydrochloride | FK-1160,NTA-194,FK 1160,FK1160,tiaramide | Others |
Tiaramide hydrochloride (FK-1160) is an anti-inflammatory drug that inhibits the action of mediators released from mast cells and has direct smooth muscle relaxant properties. | |||
T8826 | 3-AMINO-1,2,4-TRIAZINE | Others | |
3-AMINO-1,2,4-TRIAZINE is an aromatic bioactive compound. It has been used to synthesize a variety of drugs, including the antifungal drug fluconazole, the anti-inflammatory drug ibuprofen and the anticancer drug paclita... | |||
T2553 | Etofenamate | COX | |
Etofenamate is a non-steroidal anti-inflammatory drug (NSAID) used for the treatment of joint and muscular pain. | |||
T5843 | Tarenflurbil | MPC7869,(R)-Flurbiprofen,R-flurbiprofen | Retinoid Receptor , Autophagy |
Tarenflurbil ((R)-Flurbiprofen) is the non-cyclooxygenase inhibiting R-enantiomer of the non-steroidal anti-inflammatory drug flurbiprofen, which was assessed as a remedy for Alzheimer's disease. | |||
T7207 | FK 3311 | FK-3311,COX-2 Inhibitor V | COX |
FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (NSAID) | |||
T0435 | Sulfinpyrazone | (+/-)-Sulfinpyrazone,G-28315,NSC 75925 | COX |
Sulfinpyrazone (NSC-75925) is a uricosuric drug that is used to reduce the serum urate levels in gout therapy. It lacks anti-inflammatory, analgesic, and diuretic properties. | |||
T0484 | Deracoxib | SC 46,SC 046,SC 59046 | Apoptosis , COX |
Deracoxib (SC 46) is a non-steroidal, non-narcotic anti-inflammatory drug. It is also a selective cyclooxygenase-2 inhibitor, and IC50 Value: 70 to 150 μM(inhibition of 3 osteosarcoma cell lines). | |||
T0458 | Indomethacin | Indocin,Indometacine,Indomethacine,Indometacin | Phospholipase , COX , PDE , Autophagy |
Indomethacin (Indometacin) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of indomethacin is as a Cyclooxygenase Inhibitor. |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T1468 | Lornoxicam | Ro 13-9297,Chlortenoxicam,TS110 | COX , Endogenous Metabolite |
Lornoxicam (Chlortenoxicam) (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory, and antipyretic properties. Lornoxicam differs from other oxicam co... | |||
T2959 | Ginsenoside Rh2 | 20(S)-Rh2,20S-Ginsenoside Rh2,20(S)-Ginsenoside Rh2 | Apoptosis , EGFR , Caspase , Endogenous Metabolite |
Ginsenoside Rh2 (20(S)-Ginsenoside Rh2), an extract of red Panax ginseng, is a potent anti-inflammatory and anticancer drug. | |||
T6S1683 | Demethoxycurcumin | Curcumin II,Desmethoxycurcumin,Monodemethoxycurcumin | Apoptosis , Antioxidant , Antibacterial , Autophagy |
1. Demethoxycurcumin (Desmethoxycurcumin) has antioxidant activity. 2. Demethoxycurcumin has anti-inflammatory activity. 3. Demethoxycurcumin has anti-proliferative activity. 4. Demethoxycurcumin has anti-acanthamoebic e... | |||
T6926 | Palmitoylethanolamide | Mackpeart DR 14V,N-palmitoylethanolamine,Loramine P 256,Impulsin,AM 3112,Palmidrol | Influenza Virus , Endogenous Metabolite , PPAR |
Palmitoylethanolamide (Impulsin) is an endogenously fatty acid amide. It has a role as an anti-inflammatory drug, an antihypertensive agent, a neuroprotective agent and an anticonvulsant.Upon administration, palmitoyleth... | |||
T2787 | Picroside I | 6'-Cinnamoylcatalpol | MMP , STAT |
Picroside I (6'-Cinnamoylcatalpol), a hepatoprotective agent, is reported to be antimicrobial and used against hepatitis B. It has antioxidant, and anti-inflammatory activities, it may be the valuable anti-invasive drug ... | |||
T3S2296 | Gardenoside | Others | |
Gardenoside has hepatoprotective, pain‑relieving, and anti-mastitis effects. it may be a potential therapeutic herb against NASH by suppressed supernatant inflammatory cytokine production and intracellular NFkB act... | |||
T3S1471 | Cucurbitacin IIA | Dihydrocucurbitacin Q1,Hemslecin A,Curcurbitacin IIA | Apoptosis , Survivin |
1. Cucurbitacin IIA (Dihydrocucurbitacin Q1) can induce apoptosis and enhance autophagy , contributes to the anti-inflammatory activity of Cucurbitacin IIA against inflammation-related diseases. 2. Cucurbitacin IIA is a ... | |||
T4518 | Licochalcone D | ERK , NF-κB | |
Licochalcone D may be a potential drug for human melanoma treatment by inhibiting proliferation, inducing apoptosis via the mitochondrial pathway and blocking cell migration and invasion. Licochalcone D has cardioprotect... | |||
T4S1962 | Beta-Asarone | Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin | NF-κB , JNK |
1. beta-Asarone (Cis-Isoelemicin) may be a potential preventive drug for Alzheimer's disease. 2. Beta-Asarone prevents autophagy and synaptic loss by reducing ROCK expression in SAMP8 mice. 3. The co-administration of be... | |||
T10619 | Bromelain | Apoptosis , Others | |
Bromelain is an anti-inflammatory drug derived from pineapple stem. It acts through down-regulation of plasma kininogen, degradation of advanced glycation end-product receptors, inhibition of Prostaglandin E2 expression,... | |||
T3794 | Pentagalloylglucose | Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose | Influenza Virus |
1, 2, 3, 4, 6-Pentagalloylglucose (Penta-O-galloyl-β-D-glucose) and gallic acid from Pistacia lentiscus have antimutagenic and antioxidant activities. 2. 1, 2, 3, 4, 6-Penta-O-galloyl-beta-D-glucose (PGG) possesses poten... | |||
T5S1172 | Tiliroside | Tribuloside | Antioxidant |
1. Tiliroside (Tribuloside) shows anticarcinogenic activity. 2. Tiliroside shows hepatoprotective activity. 3. Tiliroside shows antioxidant and anti-inflammatory activity, can inhibit neuroinflammation in neurodegenerati... | |||
T5S2357 | Acetylcorynoline | (+)-Corynoline Acetate,O-Acetylcorynoline | Antifungal |
1. Acetylcorynoline (O-Acetylcorynoline) has antifungal、anti-inflammatory activity. 2. Acetylcorynoline may be one of the potent immunosuppressive agents through the blockage of dendritic cells maturation and function. 3... | |||
T3417 | Amentoflavone | Didemethyl-ginkgetin,Amenthoflavone,3',8''-Biapigenin | Apoptosis , P450 , Phospholipase , Reactive Oxygen Species , Opioid Receptor , COX , Antibacterial , RSV , Antifungal |
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for drug metabolism in the body. Amentoflavone also is an inhib... | |||
T6S0077 | Byakangelicol | COX | |
1. Byakangelicol may inhibit P-gp expressed at the BBB even under in vivo conditions. 2. Byakangelicol can inhibit IL-1beta-induced PGE2 release in A549 cells; this inhibition may be mediated by suppression of COX-2 expr... | |||
T25271 | Cortivazol | Dilaster | |
Cortivazol is an Anti-Inflammatory Drug. | |||
TMA0925 | Wilforlide A acetate | Others | |
Wilforlide A (T1) serves as a quality control standard of Tripterygium Glycosides that be listed in Drug Standard of Ministry of Public Health of the People's Republic of China. T1 has anti-inflammatory effects. | |||
TN1681 | Gentianine | Others , TNF , transporter , PPAR | |
Gentianine is an effective Swertiamarin derivative, which has anti-diabetic, antipsychotic, anti-inflammatory, hypotensive, diuretic and other effects, and has the potential to be developed into a safe antihypertensive d... | |||
TN5186 | Triptoquinone A | IL Receptor , NOS | |
Triptoquinone A may be a useful candidate for the development of a drug as a potent inhibitor of iNOS gene over-expression. Triptoquinone A has anti-inflammatory activity, it prevents ndotoxin-or interleukin-1 beta-promo... | |||
TN3779 | De-O-methyllasiodiplodin | IL Receptor , TNF , ROS , Antifection | |
De-O-methyllasiodiplodin exhibits radical scavenging, moderate antibacterial, and potential anti-inflammatory effects, it shows moderate suppression effects on induced NO production. De-O-methyllasiodiplodin effectively ... | |||
TN4490 | Manassantin B | ERK , BCL , p38 MAPK , TNF , NF-κB , JNK , STAT , Antifection | |
Manassantin B is a potent inhibitor of NF-κB activation by the suppression of transciptional activity of RelA/p65 subunit of NF-κB. It also possesses anti-EBV lytic replication activity. Manassantin B inhibits interleu... | |||
T38330 | Collinin | ||
Collinin is a coumarin that has been found in Z. schinifolium and has diverse biological activities.1,2,3,4 It is active against drug-susceptible and -resistant strains of M. tuberculosis (MIC50s = 3.13-6.25 μg/ml).1 Col... |
カタログ番号 | 製品名 | Species | Expression System |
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TMPK-00759 | IgG1 Fc Protein, Human, Recombinant | Human | HEK293 Cells |
IgG1 is most abundant in serum among the four IgG subclasses (IgG1, 2, 3 and 4) and binds to Fc receptors (FcγR) on phagocytic cells with high affinity. Fc fragment is demonstrated to mediate phagocytosis, trigger inflam... | |||
TMPY-06836 | NR3C1 Protein, Human, Recombinant (His) | Human | E. coli |
NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene. This gene encodes glucocorticoid receptor, which can function both as a transcription factor that binds to glucocorticoid response elements ... | |||
TMPJ-00751 | IgG4 hFc Protein, Human, Recombinant (aa 99-326) | Human | HEK293 Cells |
As a monomeric immunoglobulin that is predominately involved in the secondary antibody response and the only isotype that can pass through the human placenta, Immunoglobulin G (IgG) is synthesized and secreted by plasma ... |
カタログ番号 | 製品名 | ||
---|---|---|---|
L4710 | Nonsteroidal Anti-Inflammatory Compound Library | 530 compounds | |
530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening. | |||
L6710 | Anti-Inflammatory Traditional Chinese Medicine Compound Library | 1246 compounds | |
A collection of 1246 TCM monomers with anti-inflammatory activity or targeting molecular therapeutic targets in inflammation, a powerful tool for drug discovery and mechanism study; | |||
L9810 | Anti-Fibrosis Compound Library | 1180 compounds | |
A unique collection of 1180 potential anti-fibrosis compounds, can be used in HTS and HCS; | |||
L4700 | Immunology/Inflammation Compound Library | 4720 compounds | |
A unique collection of 4720 anti-inflammation compounds effective for high throughput screening and high content screening. | |||
L6110 | Alkaloid Natural Product Library | 464 compounds | |
A unique collection of 464 natural alkaloids can be used for high throughput and high content screening; | |||
L6100 | Polyphenolic Natural Product Library | 635 compounds | |
A unique collection of 635 natural polyphenolic compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L6810 | Traditional Chinese Medicine Monomer Library | 2755 compounds | |
A unique collection of 2755 compounds (TCM monomers) sourcing from traditional Chinese Medicines, is a powerful tool for drug discovery and research in mechanism; | |||
L9610 | Cyclic Peptide Library | 55 compounds | |
55 species of cyclic peptide molecules for high-throughput and high-content screening; | |||
L6730 | Anti-virus Traditional Chinese Medicine Monomer Library | 268 compounds | |
A collection of 268 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies. | |||
L9000 | Apoptosis Compound Library | 1760 compounds | |
A unique collection of 1760 apoptosis-related compounds for apoptosis research, research in tumorigenesis, and anti-cancer drug screening; | |||
L6400 | Marine Natural Product Library | 144 compounds | |
A unique collection of 144 marine natural products for high throughput screening (HTS) and high content screening (HCS); | |||
L5100 | Fluorochemical Library | 574 compounds | |
A unique collection of 574 fluorochemicals that can be used for high through-put screening (HTS) and high content screening (HCS); | |||
L6820 | Tobacco Monomer Library | 747 compounds | |